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5-HT receptor

Index 5-HT receptor

5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in the central and peripheral nervous systems. [1]

Table of Contents

  1. 241 relations: A-372159, Acetylcholine, Adrenaline, Adrenergic receptor, Adrenocorticotropic hormone, Agomelatine, Agonist, AL-38022A, Almotriptan, Alosetron, Alprenolol, Amitriptyline, Analgesic, Anorectic, Antidepressant, Antiemetic, Antihypertensive drug, Antimigraine drug, Antipsychotic, Anxiety, Anxiolytic, Appetite stimulant, AR-A000002, Aripiprazole, AS-19 (drug), Asenapine, Atypical antipsychotic, Autoreceptor, Benzylpiperazine, BIMU8, Blood vessel, BMY-7378, BRL-15,572, BRL-54443, Bryan Roth, Bufotenin, Buspirone, BW-723C86, Caenorhabditis elegans, Cell membrane, Central nervous system, CGS-12066A, Cinitapride, Cisapride, Clomipramine, Cloning, Clozapine, Cognition, Cortisol, CP-135807, ... Expand index (191 more) »

  2. Serotonin receptors

A-372159

A-372159 is a drug which acts as a potent and selective partial agonist for the 5HT2C receptor, with more than 100x selectivity over the closely related 5-HT2B receptor and a Ki of 3nM.

See 5-HT receptor and A-372159

Acetylcholine

Acetylcholine (ACh) is an organic compound that functions in the brain and body of many types of animals (including humans) as a neurotransmitter.

See 5-HT receptor and Acetylcholine

Adrenaline

Adrenaline, also known as epinephrine, is a hormone and medication which is involved in regulating visceral functions (e.g., respiration).

See 5-HT receptor and Adrenaline

Adrenergic receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, beta-2 (β2) agonists and alpha-2 (α2) agonists, which are used to treat high blood pressure and asthma, for example.

See 5-HT receptor and Adrenergic receptor

Adrenocorticotropic hormone

Adrenocorticotropic hormone (ACTH; also adrenocorticotropin, corticotropin) is a polypeptide tropic hormone produced by and secreted by the anterior pituitary gland.

See 5-HT receptor and Adrenocorticotropic hormone

Agomelatine

Agomelatine, sold under the brand names Valdoxan and Thymanax, among others, is an atypical antidepressant most commonly used to treat major depressive disorder and generalized anxiety disorder.

See 5-HT receptor and Agomelatine

Agonist

An agonist is a chemical that activates a receptor to produce a biological response.

See 5-HT receptor and Agonist

AL-38022A

AL-38022A is an indazole derivative drug which is one of a range of similar drugs developed for scientific research and with some possible clinical applications.

See 5-HT receptor and AL-38022A

Almotriptan

Almotriptan (trade name Axert and others) is a triptan medication discovered and developed by Almirall for the treatment of heavy migraine headache.

See 5-HT receptor and Almotriptan

Alosetron

Alosetron, sold under the brand name Lotronex among others, is a 5-HT3 antagonist used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in females only.

See 5-HT receptor and Alosetron

Alprenolol

Alprenolol, or alfeprol, alpheprol, and alprenololum (Gubernal, Regletin, Yobir, Apllobal, Aptine, Aptol Duriles), is a non-selective beta blocker as well as a 5-HT1A and 5-HT1B receptor antagonist, used in the treatment of angina pectoris.

See 5-HT receptor and Alprenolol

Amitriptyline

Amitriptyline, sold under the brand name Elavil among others, is a tricyclic antidepressant primarily used to treat major depressive disorder, and a variety of pain syndromes such as neuropathic pain, fibromyalgia, migraine and tension headaches.

See 5-HT receptor and Amitriptyline

Analgesic

An analgesic drug, also called simply an analgesic, antalgic, pain reliever, or painkiller, is any member of the group of drugs used for pain management.

See 5-HT receptor and Analgesic

Anorectic

An anorectic or anorexic is a drug which reduces appetite, resulting in lower food consumption, leading to weight loss.

See 5-HT receptor and Anorectic

Antidepressant

Antidepressants are a class of medications used to treat major depressive disorder, anxiety disorders, chronic pain, and addiction.

See 5-HT receptor and Antidepressant

Antiemetic

An antiemetic is a drug that is effective against vomiting and nausea.

See 5-HT receptor and Antiemetic

Antihypertensive drug

Antihypertensives are a class of drugs that are used to treat hypertension (high blood pressure).

See 5-HT receptor and Antihypertensive drug

Antimigraine drug

Antimigraine drugs are medications intended to reduce the effects or intensity of migraine headache.

See 5-HT receptor and Antimigraine drug

Antipsychotic

Antipsychotics, previously known as neuroleptics and major tranquilizers, are a class of psychotropic medication primarily used to manage psychosis (including delusions, hallucinations, paranoia or disordered thought), principally in schizophrenia but also in a range of other psychotic disorders.

See 5-HT receptor and Antipsychotic

Anxiety

Anxiety is an emotion which is characterised by an unpleasant state of inner turmoil and includes feelings of dread over anticipated events.

See 5-HT receptor and Anxiety

Anxiolytic

An anxiolytic (also antipanic or anti-anxiety agent) is a medication or other intervention that reduces anxiety.

See 5-HT receptor and Anxiolytic

Appetite stimulant

An orexigenic, or appetite stimulant, is a drug, hormone, or compound that increases appetite and may induce hyperphagia.

See 5-HT receptor and Appetite stimulant

AR-A000002

AR-A000002 is a drug which is one of the first compounds developed to act as a selective antagonist for the serotonin receptor 5-HT1B, with approximately 10x selectivity for 5-HT1B over the closely related 5-HT1D receptor.

See 5-HT receptor and AR-A000002

Aripiprazole

Aripiprazole, sold under the brand names Abilify and Aristada, among others, is an atypical antipsychotic. It is primarily used in the treatment of schizophrenia and bipolar disorder; other uses include as an add-on treatment in major depressive disorder and obsessive compulsive disorder (OCD), tic disorders, and irritability associated with autism.

See 5-HT receptor and Aripiprazole

AS-19 (drug)

AS-19 is a substance which acts as a potent agonist at the 5-HT7 receptor, with an IC50 of 0.83 nM.

See 5-HT receptor and AS-19 (drug)

Asenapine

Asenapine, sold under the brand name Saphris among others, is an atypical antipsychotic medication used to treat schizophrenia and acute mania associated with bipolar disorder as well as the medium to long-term management of bipolar disorder.

See 5-HT receptor and Asenapine

Atypical antipsychotic

The atypical antipsychotics (AAP), also known as second generation antipsychotics (SGAs) and serotonin–dopamine antagonists (SDAs), are a group of antipsychotic drugs (antipsychotic drugs in general are also known as tranquilizers and neuroleptics, although the latter is usually reserved for the typical antipsychotics) largely introduced after the 1970s and used to treat psychiatric conditions.

See 5-HT receptor and Atypical antipsychotic

Autoreceptor

An autoreceptor is a type of receptor located in the membranes of nerve cells.

See 5-HT receptor and Autoreceptor

Benzylpiperazine

Benzylpiperazine (BZP) is a substance often used as a recreational drug and is known to have euphoriant and stimulant properties.

See 5-HT receptor and Benzylpiperazine

BIMU8

BIMU-8 is a drug which acts as a 5-HT4 receptor selective agonist.

See 5-HT receptor and BIMU8

Blood vessel

Blood vessels are the structures of the circulatory system that transport blood throughout the human body.

See 5-HT receptor and Blood vessel

BMY-7378

BMY-7,378 is a 5-HT1A receptor weak partial agonist/antagonist and α1D-adrenergic receptor antagonist.

See 5-HT receptor and BMY-7378

BRL-15,572

BRL-15,572 is a drug which acts as a selective antagonist for the serotonin receptor subtype 5-HT1D, with around 60x selectivity over other related receptors.

See 5-HT receptor and BRL-15,572

BRL-54443

BRL-54443 is a drug which acts as a selective agonist for the 5-HT1E and 5-HT1F serotonin receptor subtypes.

See 5-HT receptor and BRL-54443

Bryan Roth

Bryan L. Roth is the Michael Hooker Distinguished Professor of Protein Therapeutics and Translational Proteomics, UNC School of Medicine.

See 5-HT receptor and Bryan Roth

Bufotenin

Bufotenin (5-HO-DMT, bufotenine, dimethylserotonin) is a tryptamine derivative, more specifically, a DMT analog, related to the neurotransmitter serotonin.

See 5-HT receptor and Bufotenin

Buspirone

Buspirone, sold under the brand name Buspar, among others, is an anxiolytic, a medication primarily used to treat anxiety disorders, particularly generalized anxiety disorder.

See 5-HT receptor and Buspirone

BW-723C86

BW-723C86 is a tryptamine derivative drug which acts as a 5-HT2B receptor agonist.

See 5-HT receptor and BW-723C86

Caenorhabditis elegans

Caenorhabditis elegans is a free-living transparent nematode about 1 mm in length that lives in temperate soil environments.

See 5-HT receptor and Caenorhabditis elegans

Cell membrane

The cell membrane (also known as the plasma membrane or cytoplasmic membrane, and historically referred to as the plasmalemma) is a biological membrane that separates and protects the interior of a cell from the outside environment (the extracellular space).

See 5-HT receptor and Cell membrane

Central nervous system

The central nervous system (CNS) is the part of the nervous system consisting primarily of the brain and spinal cord.

See 5-HT receptor and Central nervous system

CGS-12066A

CGS-12066A is a drug which acts as a potent and selective agonist for the 5-HT1B receptor with lower affinity for the three 5-HT2 receptor subtypes.

See 5-HT receptor and CGS-12066A

Cinitapride

Cinitapride (trade names Cintapro, Pemix) is a gastroprokinetic agent and antiemetic agent of the benzamide class which is marketed in India, Mexico, Pakistan and Spain.

See 5-HT receptor and Cinitapride

Cisapride

Cisapride is a gastroprokinetic agent, a drug that increases motility in the upper gastrointestinal tract.

See 5-HT receptor and Cisapride

Clomipramine

Clomipramine, sold under the brand name Anafranil among others, is a tricyclic antidepressant (TCA).

See 5-HT receptor and Clomipramine

Cloning

Cloning is the process of producing individual organisms with identical genomes, either by natural or artificial means.

See 5-HT receptor and Cloning

Clozapine

Clozapine is a psychiatric medication and was the first atypical antipsychotic (also called second-generation antipsychotic) to be discovered.

See 5-HT receptor and Clozapine

Cognition

Cognition is the "mental action or process of acquiring knowledge and understanding through thought, experience, and the senses".

See 5-HT receptor and Cognition

Cortisol

Cortisol is a steroid hormone in the glucocorticoid class of hormones and a stress hormone.

See 5-HT receptor and Cortisol

CP-135807

CP-135807 is a drug which acts as a potent and selective agonist for the 5-HT1D serotonin receptor, and is used to study the function of this receptor subtype.

See 5-HT receptor and CP-135807

CP-93129

CP-93129 is a drug which acts as a potent and selective serotonin 5-HT1B receptor agonist, with approximately 150x and 200x selectivity over the closely related 5-HT1D and 5-HT1A receptors.

See 5-HT receptor and CP-93129

CP-94253

CP-94253 is a drug which acts as a potent and selective serotonin 5-HT1B receptor agonist, with approximately 25× and 40× selectivity over the closely related 5-HT1D and 5-HT1A receptors.

See 5-HT receptor and CP-94253

Cyanopindolol

Cyanopindolol is a drug related to pindolol which acts as both a β1 adrenoceptor antagonist and a 5-HT1A receptor antagonist.

See 5-HT receptor and Cyanopindolol

Cyclic adenosine monophosphate

Cyclic adenosine monophosphate (cAMP, cyclic AMP, or 3',5'-cyclic adenosine monophosphate) is a second messenger, or cellular signal occurring within cells, that is important in many biological processes.

See 5-HT receptor and Cyclic adenosine monophosphate

Cyproheptadine

Cyproheptadine, sold under the brand name Periactin among others, is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties.

See 5-HT receptor and Cyproheptadine

Dazopride

Dazopride (AHR-5531) is an antiemetic and gastroprokinetic agent of the benzamide class which was never marketed.

See 5-HT receptor and Dazopride

Depolarization

In biology, depolarization or hypopolarization is a change within a cell, during which the cell undergoes a shift in electric charge distribution, resulting in less negative charge inside the cell compared to the outside.

See 5-HT receptor and Depolarization

Diglyceride

A diglyceride, or diacylglycerol (DAG), is a glyceride consisting of two fatty acid chains covalently bonded to a glycerol molecule through ester linkages.

See 5-HT receptor and Diglyceride

Dihydroergotamine

Dihydroergotamine (DHE), sold under the brand names D.H.E. 45 and Migranal among others, is an ergot alkaloid used to treat migraines.

See 5-HT receptor and Dihydroergotamine

Dolasetron

Dolasetron (trade name Anzemet) is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy.

See 5-HT receptor and Dolasetron

Dopamine

Dopamine (DA, a contraction of 3,4-dihydroxyphenethylamine) is a neuromodulatory molecule that plays several important roles in cells.

See 5-HT receptor and Dopamine

Doxepin

Doxepin is a medication belonging to the tricyclic antidepressant (TCA) class of drugs used to treat major depressive disorder, anxiety disorders, chronic hives, and insomnia.

See 5-HT receptor and Doxepin

E-55888

E-55888 is a drug developed by Esteve, which acts as a potent and selective full agonist at the 5HT7 serotonin receptor, and is used for investigating the role of 5-HT7 receptors in the perception of pain.

See 5-HT receptor and E-55888

E-6837

E-6837 is an orally active, 5-HT6 agonist developed in an attempt to create an anti-obesity medication.

See 5-HT receptor and E-6837

EGIS-12,233

EGIS-12,233 is a drug with applications in scientific research, acting as a potent and selective antagonist for both the 5-HT6 and 5-HT7 serotonin receptor subtypes, with good selectivity over other receptors.

See 5-HT receptor and EGIS-12,233

Eletriptan

Eletriptan, sold under the brand name Relpax and used in the form of eletriptan hydrobromide, is a second-generation triptan medication intended for treatment of migraine headaches.

See 5-HT receptor and Eletriptan

Eltoprazine

Eltoprazine (developmental code name DU-28,853) is a serotonergic drug of the phenylpiperazine class which is described as a serenic or antiaggressive agent.

See 5-HT receptor and Eltoprazine

EMD-386088

EMD-386088 is an indole derivative which is used in scientific research.

See 5-HT receptor and EMD-386088

EMDT

2-Ethyl-5-methoxy-N,N-dimethyltryptamine (EMDT) is a tryptamine derivative which is used in scientific research.

See 5-HT receptor and EMDT

Empathogen

Empathogens or entactogens are a class of psychoactive drugs that induce the production of experiences of emotional communion, oneness, relatedness, emotional openness—that is, empathy or sympathy—as particularly observed and reported for experiences with 3,4-methylenedioxymethamphetamine (MDMA).

See 5-HT receptor and Empathogen

Eplivanserin

Eplivanserin (SR-46,349; planned trade name Ciltyri) was an experimental drug for the treatment of insomnia which was being developed by Sanofi Aventis.

See 5-HT receptor and Eplivanserin

Ergometrine

Ergometrine, also known as ergonovine and sold under the brand names Ergotrate, Ergostat, and Syntometrine among others, is a medication used to cause contractions of the uterus to treat heavy vaginal bleeding after childbirth.

See 5-HT receptor and Ergometrine

Ergotamine

Ergotamine, sold under the brand name Ergomar among others, is an ergopeptine and part of the ergot family of alkaloids; it is structurally and biochemically closely related to ergoline.

See 5-HT receptor and Ergotamine

Etoperidone

Etoperidone, associated with several brand names, is an atypical antidepressant which was developed in the 1970s and either is no longer marketed or was never marketed.

See 5-HT receptor and Etoperidone

F-15,599

F-15,599, also known as NLX-101, is a potent and selective 5-HT1A receptor full agonist.

See 5-HT receptor and F-15,599

Fenfluramine

Fenfluramine, sold under the brand name Fintepla, is a serotonergic medication used for the treatment of seizures associated with Dravet syndrome and Lennox–Gastaut syndrome.

See 5-HT receptor and Fenfluramine

Flesinoxan

Flesinoxan (DU-29,373) is a potent and selective 5-HT1A receptor partial/near-full agonist of the phenylpiperazine class.

See 5-HT receptor and Flesinoxan

Fluoxetine

Fluoxetine, sold under the brand name Prozac, among others, is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class.

See 5-HT receptor and Fluoxetine

Frovatriptan

Frovatriptan, sold under the brand name Frova, is a triptan drug developed by Vernalis for the treatment of migraine headaches and for short term prevention of menstrual migraine.

See 5-HT receptor and Frovatriptan

G protein-coupled receptor

G protein-coupled receptors (GPCRs), also known as seven-(pass)-transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptors, and G protein-linked receptors (GPLR), form a large group of evolutionarily related proteins that are cell surface receptors that detect molecules outside the cell and activate cellular responses.

See 5-HT receptor and G protein-coupled receptor

GABA

GABA (gamma Aminobutyric acid, γ-Aminobutyric acid) is the chief inhibitory neurotransmitter in the developmentally mature mammalian central nervous system.

See 5-HT receptor and GABA

Gastrointestinal tract

The gastrointestinal tract (GI tract, digestive tract, alimentary canal) is the tract or passageway of the digestive system that leads from the mouth to the anus. The GI tract contains all the major organs of the digestive system, in humans and other animals, including the esophagus, stomach, and intestines.

See 5-HT receptor and Gastrointestinal tract

Gepirone

Gepirone, sold under the brand name Exxua, is a medication used for the treatment of major depressive disorder.

See 5-HT receptor and Gepirone

Gi alpha subunit

Gi protein alpha subunit is a family of heterotrimeric G protein alpha subunits.

See 5-HT receptor and Gi alpha subunit

Glossary of biology

This glossary of biology terms is a list of definitions of fundamental terms and concepts used in biology, the study of life and of living organisms.

See 5-HT receptor and Glossary of biology

Glutamic acid

Glutamic acid (symbol Glu or E; the anionic form is known as glutamate) is an α-amino acid that is used by almost all living beings in the biosynthesis of proteins.

See 5-HT receptor and Glutamic acid

Gq alpha subunit

Gq protein alpha subunit is a family of heterotrimeric G protein alpha subunits.

See 5-HT receptor and Gq alpha subunit

GR-127935

GR-127935 is a drug which acts as a selective antagonist at the serotonin receptors 5-HT1B and 5-HT1D.

See 5-HT receptor and GR-127935

Granisetron

Granisetron is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy and radiotherapy.

See 5-HT receptor and Granisetron

Gs alpha subunit

The Gs alpha subunit (Gαs, Gsα) is a subunit of the heterotrimeric G protein Gs that stimulates the cAMP-dependent pathway by activating adenylyl cyclase.

See 5-HT receptor and Gs alpha subunit

Hallucinogen

Hallucinogens are a large and diverse class of psychoactive drugs that can produce altered states of consciousness characterized by major alterations in thought, mood, and perception as well as other changes.

See 5-HT receptor and Hallucinogen

Haloperidol

Haloperidol, sold under the brand name Haldol among others, is a typical antipsychotic medication.

See 5-HT receptor and Haloperidol

Heteroreceptor

A heteroreceptor is a receptor regulating the synthesis and/or the release of mediators other than its own ligand.

See 5-HT receptor and Heteroreceptor

Hydroxyzine

Hydroxyzine, sold under the brand names Atarax and Vistaril among others, is an antihistamine medication.

See 5-HT receptor and Hydroxyzine

Hypnotic

Hypnotic (from Greek Hypnos, sleep), or soporific drugs, commonly known as sleeping pills, are a class of (and umbrella term for) psychoactive drugs whose primary function is to induce sleep (or surgical anesthesiaWhen used in anesthesia to produce and maintain unconsciousness, "sleep" is metaphorical as there are no regular sleep stages or cyclical natural states; patients rarely recover from anesthesia feeling refreshed and with renewed energy.

See 5-HT receptor and Hypnotic

Iloperidone

Iloperidone, commonly known as Fanapt and previously known as Zomaril, is an atypical antipsychotic for the treatment of schizophrenia.

See 5-HT receptor and Iloperidone

Imipramine

Imipramine, sold under the brand name Tofranil, among others, is a tricyclic antidepressant (TCA) mainly used in the treatment of depression.

See 5-HT receptor and Imipramine

Inositol trisphosphate

Inositol trisphosphate or inositol 1,4,5-trisphosphate abbreviated InsP3 or Ins3P or IP3 is an inositol phosphate signaling molecule.

See 5-HT receptor and Inositol trisphosphate

Iodocyanopindolol

Iodocyanopindolol (INN) is a drug related to pindolol which acts as both a β1 adrenoreceptor antagonist and a 5-HT1A receptor antagonist.

See 5-HT receptor and Iodocyanopindolol

Ion channel

Ion channels are pore-forming membrane proteins that allow ions to pass through the channel pore.

See 5-HT receptor and Ion channel

Ipsapirone

Ipsapirone is a selective 5-HT1A receptor partial agonist of the piperazine and azapirone chemical classes.

See 5-HT receptor and Ipsapirone

Isamoltane

Isamoltane (CGP-361A) is a drug used in scientific research.

See 5-HT receptor and Isamoltane

Ketanserin

Ketanserin (INN, USAN, BAN) (brand name Sufrexal; former developmental code name R41468) is a drug used clinically as an antihypertensive agent and in scientific research to study the serotonergic system; specifically, the 5-HT2 receptor family. It was discovered at Janssen Pharmaceutica in 1980. It is not available in the United States.

See 5-HT receptor and Ketanserin

Lasmiditan

Lasmiditan, sold under the brand name Reyvow, is a medication used for the acute (active but short-term) treatment of migraine with or without aura (a sensory phenomenon or visual disturbance) in adults.

See 5-HT receptor and Lasmiditan

Latrepirdine

Latrepirdine (INN, also known as dimebolin and sold as Dimebon) is an antihistamine drug which has been used clinically in Russia since 1983.

See 5-HT receptor and Latrepirdine

Lecozotan

Lecozotan is an investigational drug by Wyeth tested for improvement of cognitive functions of Alzheimer's disease patients.

See 5-HT receptor and Lecozotan

Ligand (biochemistry)

In biochemistry and pharmacology, a ligand is a substance that forms a complex with a biomolecule to serve a biological purpose.

See 5-HT receptor and Ligand (biochemistry)

Ligand-gated ion channel

Ligand-gated ion channels (LICs, LGIC), also commonly referred to as ionotropic receptors, are a group of transmembrane ion-channel proteins which open to allow ions such as Na+, K+, Ca2+, and/or Cl− to pass through the membrane in response to the binding of a chemical messenger (i.e. a ligand), such as a neurotransmitter.

See 5-HT receptor and Ligand-gated ion channel

Lisuride

Lisuride, sold under the brand name Dopergin among others, is a monoaminergic medication of the ergoline class which is used in the treatment of Parkinson's disease, migraine, and high prolactin levels.

See 5-HT receptor and Lisuride

Lorcaserin

Lorcaserin, marketed under the brand name Belviq, was a weight-loss drug developed by Arena Pharmaceuticals.

See 5-HT receptor and Lorcaserin

LSD

Lysergic acid diethylamide, commonly known as LSD (from German Lysergsäure-diethylamid), and known colloquially as acid or lucy, is a potent psychedelic drug.

See 5-HT receptor and LSD

LY-334370

LY-334370 is a selective 5-HT1F receptor agonist which was under development by Eli Lilly and Company for the treatment of migraine headaches.

See 5-HT receptor and LY-334370

Lysine

Lysine (symbol Lys or K) is an α-amino acid that is a precursor to many proteins.

See 5-HT receptor and Lysine

MDMA

3,4-Methylenedioxymethamphetamine (MDMA), commonly known as ecstasy (tablet form), and molly or mandy (crystal form), is a potent empathogen–entactogen with stimulant and minor psychedelic properties.

See 5-HT receptor and MDMA

Mefway (18F)

Mefway is a serotonin 5-HT1A receptor antagonist used in medical research, usually in the form of mefway (18F) as a positron emission tomography (PET) radiotracer.

See 5-HT receptor and Mefway (18F)

Memantine

Memantine, sold under the brand name Axura among others, is a medication used to slow the progression of moderate-to-severe Alzheimer's disease. It is taken by mouth. Common side effects include headache, constipation, sleepiness, and dizziness. Severe side effects may include blood clots, psychosis, and heart failure.

See 5-HT receptor and Memantine

Mescaline

Mescaline or mescalin (3,4,5-trimethoxyphenethylamine) is a naturally occurring psychedelic protoalkaloid of the substituted phenethylamine class, known for its hallucinogenic effects comparable to those of LSD and psilocybin.

See 5-HT receptor and Mescaline

Metergoline

Metergoline, also known as methergoline and sold under the brand names Contralac (veterinary) and Liserdol (clinical), is a monoaminergic medication of the ergoline group which is used as a prolactin inhibitor in the treatment of hyperprolactinemia (high prolactin levels) and to suppress lactation.

See 5-HT receptor and Metergoline

Methylergometrine

Methylergometrine, also known as methylergonovine and sold under the brand name Methergine, is a medication of the ergoline and lysergamide groups which is used as an oxytocic in obstetrics and in the treatment of migraine.

See 5-HT receptor and Methylergometrine

Methylphenidate

Methylphenidate, sold under the brand names Ritalin and Concerta among others, is a potent central nervous system (CNS) stimulant used medically to treat attention deficit hyperactivity disorder (ADHD) and, to a lesser extent, narcolepsy.

See 5-HT receptor and Methylphenidate

Methysergide

Methysergide, sold under the brand names Deseril and Sansert, is a monoaminergic medication of the ergoline and lysergamide groups which is used in the prophylaxis and treatment of migraine and cluster headaches.

See 5-HT receptor and Methysergide

Metitepine

Metitepine (developmental code names Ro 8-6837 (maleate), VUFB-6276 (mesylate)), also known as methiothepin, is a drug described as a "psychotropic agent" of the tricyclic group which was never marketed.

See 5-HT receptor and Metitepine

Metoclopramide

Metoclopramide is a medication used for stomach and esophageal problems.

See 5-HT receptor and Metoclopramide

Mianserin

Mianserin, sold under the brand name Tolvon among others, is an atypical antidepressant that is used primarily in the treatment of depression in Europe and elsewhere in the world.

See 5-HT receptor and Mianserin

Migraine

Migraine is a genetically influenced complex neurological disorder characterized by episodes of moderate-to-severe headache, most often unilateral and generally associated with nausea and light and sound sensitivity.

See 5-HT receptor and Migraine

Mirtazapine

Mirtazapine, sold under the brand name Remeron among others, is an atypical tetracyclic antidepressant, and as such is used primarily to treat depression.

See 5-HT receptor and Mirtazapine

Mood (psychology)

In psychology, a mood is an affective state.

See 5-HT receptor and Mood (psychology)

Mosapride

Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist.

See 5-HT receptor and Mosapride

MS-245

MS-245 is a tryptamine derivative used in scientific research.

See 5-HT receptor and MS-245

NAN-190

NAN-190 is a drug and research chemical widely used in scientific studies.

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Naratriptan

Naratriptan (trade names include Amerge) is a triptan drug marketed by GlaxoSmithKline and is used for the treatment of migraine headaches.

See 5-HT receptor and Naratriptan

Nebivolol

Nebivolol is a beta blocker used to treat high blood pressure and heart failure.

See 5-HT receptor and Nebivolol

Nefazodone

Nefazodone, sold formerly under the brand names Serzone, Dutonin, and Nefadar among others, is an atypical antidepressant medication which is used in the treatment of depression and for other uses.

See 5-HT receptor and Nefazodone

Nematode

The nematodes (or; Νηματώδη; Nematoda), roundworms or eelworms constitute the phylum Nematoda.

See 5-HT receptor and Nematode

Neurotransmission

Neurotransmission (Latin: transmissio "passage, crossing" from transmittere "send, let through") is the process by which signaling molecules called neurotransmitters are released by the axon terminal of a neuron (the presynaptic neuron), and bind to and react with the receptors on the dendrites of another neuron (the postsynaptic neuron) a short distance away.

See 5-HT receptor and Neurotransmission

Neurotransmitter

A neurotransmitter is a signaling molecule secreted by a neuron to affect another cell across a synapse.

See 5-HT receptor and Neurotransmitter

Nootropic

Nootropics (or; but not or, which are common mispronunciations), colloquially brain supplements, smart drugs and cognitive enhancers, are natural, semisynthetic or synthetic compounds which purportedly improve cognitive functions, such as executive functions, attention or memory.

See 5-HT receptor and Nootropic

Noradrenergic and specific serotonergic antidepressant

Noradrenergic and specific serotonergic antidepressants (NaSSAs) are a class of psychiatric drugs used primarily as antidepressants.

See 5-HT receptor and Noradrenergic and specific serotonergic antidepressant

Norepinephrine

Norepinephrine (NE), also called noradrenaline (NA) or noradrenalin, is an organic chemical in the catecholamine family that functions in the brain and body as a hormone, neurotransmitter and neuromodulator.

See 5-HT receptor and Norepinephrine

Norfenfluramine

Norfenfluramine, or 3-trifluoromethylamphetamine, is a never-marketed drug of the amphetamine family that behaves as a serotonin and norepinephrine releasing agent and potent 5-HT2A, 5-HT2B, and 5-HT2C agonist.

See 5-HT receptor and Norfenfluramine

Olanzapine

Olanzapine, sold under the brand name Zyprexa among others, is an atypical antipsychotic primarily used to treat schizophrenia and bipolar disorder.

See 5-HT receptor and Olanzapine

Ondansetron

Ondansetron, sold under the brand name Zofran among others, is a medication used to prevent nausea and vomiting caused by cancer chemotherapy, radiation therapy, migraines or surgery.

See 5-HT receptor and Ondansetron

Oxprenolol

Oxprenolol (brand names Trasacor, Trasicor, Coretal, Laracor, Slow-Pren, Captol, Corbeton, Slow-Trasicor, Tevacor, Trasitensin, Trasidex) is a non-selective beta blocker with some intrinsic sympathomimetic activity.

See 5-HT receptor and Oxprenolol

Oxytocin

Oxytocin is a peptide hormone and neuropeptide normally produced in the hypothalamus and released by the posterior pituitary.

See 5-HT receptor and Oxytocin

Paroxetine

Paroxetine, sold under the brand names Paxil and Seroxat among others, is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used to treat major depressive disorder, obsessive-compulsive disorder, panic disorder, social anxiety disorder, post-traumatic stress disorder, generalized anxiety disorder, and premenstrual dysphoric disorder.

See 5-HT receptor and Paroxetine

Partial agonist

In pharmacology, partial agonists are drugs that bind to and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist.

See 5-HT receptor and Partial agonist

Peripheral nervous system

The peripheral nervous system (PNS) is one of two components that make up the nervous system of bilateral animals, with the other part being the central nervous system (CNS).

See 5-HT receptor and Peripheral nervous system

Piboserod

Piboserod is a selective 5-HT4 receptor antagonist which was marketed and manufactured by GlaxoSmithKline (GSK) under the trade name Serlipet for the management of atrial fibrillation and irritable bowel syndrome.

See 5-HT receptor and Piboserod

Pieris rapae

Pieris rapae is a small- to medium-sized butterfly species of the whites-and-yellows family Pieridae.

See 5-HT receptor and Pieris rapae

Pimavanserin

Pimavanserin, sold under the brand name Nuplazid, is an atypical antipsychotic which is approved for the treatment of Parkinson's disease psychosis and is also being studied for the treatment of Alzheimer's disease psychosis, schizophrenia, agitation, and major depressive disorder.

See 5-HT receptor and Pimavanserin

Pindolol

Pindolol, sold under the brand name Visken among others, is a nonselective beta blocker which is used in the treatment of hypertension.

See 5-HT receptor and Pindolol

Pizotifen

Pizotifen (INN) or pizotyline (USAN), trade name Sandomigran, is a benzocycloheptene-based drug used as a medicine, primarily as a preventive to reduce the frequency of recurrent migraine headaches.

See 5-HT receptor and Pizotifen

Platelet

Platelets or thrombocytes are a blood component whose function (along with the coagulation factors) is to react to bleeding from blood vessel injury by clumping, thereby initiating a blood clot.

See 5-HT receptor and Platelet

PNU-22394

PNU-22394 is a drug which acts as an agonist at serotonin 5-HT2 receptors, with strongest binding affinity for 5-HT2A and 5-HT2C and slightly weaker at 5-HT2B, although it is only a full agonist at 5-HT2C, but partial agonist at 5-HT2A and 5-HT2B.

See 5-HT receptor and PNU-22394

Potassium

Potassium is a chemical element; it has symbol K (from Neo-Latin kalium) and atomic number19.

See 5-HT receptor and Potassium

Prokinetic agent

A prokinetic agent (also prokineticin, gastroprokinetic agent, gastrokinetic agent or propulsive) is a type of small peptide drug which enhances gastrointestinal motility by increasing the frequency or strength of contractions, but without disrupting their rhythm.

See 5-HT receptor and Prokinetic agent

Prolactin

Prolactin (PRL), also known as lactotropin and mammotropin, is a protein best known for its role in enabling mammals to produce milk.

See 5-HT receptor and Prolactin

Propranolol

Propranolol, sold under the brand name Inderal among others, is a medication of the beta blocker class. It is used to treat high blood pressure, a number of types of irregular heart rate, thyrotoxicosis, capillary hemangiomas, performance anxiety, and essential tremors, as well to prevent migraine headaches, and to prevent further heart problems in those with angina or previous heart attacks.

See 5-HT receptor and Propranolol

Protein Data Bank

The Protein Data Bank (PDB) is a database for the three-dimensional structural data of large biological molecules such as proteins and nucleic acids, which is overseen by the Worldwide Protein Data Bank (wwPDB).

See 5-HT receptor and Protein Data Bank

Prucalopride

Prucalopride, sold under brand names Resolor and Motegrity among others, is a medication acting as a selective, high affinity 5-HT4 receptor agonist which targets the impaired motility associated with chronic constipation, thus normalizing bowel movements.

See 5-HT receptor and Prucalopride

Pseudogene

Pseudogenes are nonfunctional segments of DNA that resemble functional genes.

See 5-HT receptor and Pseudogene

Psilocin

Psilocin (also known as 4-HO-DMT, 4-hydroxy DMT, psilocine, psilocyn, or psilotsin) is a substituted tryptamine alkaloid and a serotonergic psychedelic substance.

See 5-HT receptor and Psilocin

Psilocybin

Psilocybin is a naturally occurring psychedelic prodrug compound produced by more than 200 species of fungi.

See 5-HT receptor and Psilocybin

Psychedelic drug

Psychedelics are a subclass of hallucinogenic drugs whose primary effect is to trigger non-ordinary mental states (known as psychedelic experiences or "trips") and a perceived "expansion of consciousness".

See 5-HT receptor and Psychedelic drug

Quetiapine

Quetiapine, sold under the brand name Seroquel among others, is an atypical antipsychotic medication used for the treatment of schizophrenia, bipolar disorder, and major depressive disorder.

See 5-HT receptor and Quetiapine

Quipazine

Quipazine is a serotonergic drug of the piperazine group which is used in scientific research.

See 5-HT receptor and Quipazine

Rauwolscine

Rauwolscine, also known as isoyohimbine, α-yohimbine, and corynanthidine, is an alkaloid found in various species within the genera Rauvolfia and Corynanthe (including Pausinystalia).

See 5-HT receptor and Rauwolscine

Receptor antagonist

A receptor antagonist is a type of receptor ligand or drug that blocks or dampens a biological response by binding to and blocking a receptor rather than activating it like an agonist.

See 5-HT receptor and Receptor antagonist

Renzapride

Renzapride is a prokinetic agent and antiemetic which acts as a full 5-HT4 agonist and partial 5-HT3 antagonist.

See 5-HT receptor and Renzapride

Risperidone

Risperidone, sold under the brand name Risperdal among others, is an atypical antipsychotic used to treat schizophrenia and bipolar disorder.

See 5-HT receptor and Risperidone

Ritanserin

Ritanserin, also known by its developmental code name R-55667, is a serotonin antagonist medication described as an anxiolytic, antidepressant, antiparkinsonian agent, and antihypertensive agent.

See 5-HT receptor and Ritanserin

Rizatriptan

Rizatriptan, sold under the brand name Maxalt among others, is a medication used for the treatment of migraine headaches.

See 5-HT receptor and Rizatriptan

Ro 04-6790

Ro 04-6790 is a drug, developed by Hoffmann–La Roche, which has applications in scientific research.

See 5-HT receptor and Ro 04-6790

Ro60-0175

Ro60-0175 is a drug developed by Hoffmann–La Roche, which has applications in scientific research.

See 5-HT receptor and Ro60-0175

RS-127445

RS-127445 is a drug which acts as a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000 times selectivity over the closely related 5-HT2A and 5-HT2C receptors.

See 5-HT receptor and RS-127445

RS-56812

RS-56812 is a potent and selective partial agonist at the 5HT3 receptor.

See 5-HT receptor and RS-56812

RS-67,333

RS-67,333 is a drug which has been investigated as a potential rapid-acting antidepressant, nootropic, and treatment for Alzheimer's disease.

See 5-HT receptor and RS-67,333

RU-24,969

RU-24,969 is a chemical compound widely used in scientific studies.

See 5-HT receptor and RU-24,969

SB-216641

SB-216641 is a drug which is a selective antagonist for the serotonin receptor 5-HT1B, with around 25x selectivity over the closely related 5-HT1D receptor.

See 5-HT receptor and SB-216641

SB-242084

SB-242084 is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.

See 5-HT receptor and SB-242084

SB-258585

SB-258585 is a drug which is used in scientific research.

See 5-HT receptor and SB-258585

SB-269970

SB-269970 is a drug and research chemical developed by GlaxoSmithKline used in scientific studies.

See 5-HT receptor and SB-269970

SB-271046

SB-271046 is a drug which is used in scientific research.

See 5-HT receptor and SB-271046

SB-357134

SB-357134 is a drug which is used in scientific research.

See 5-HT receptor and SB-357134

SB-399885

SB-399885 is a drug which is used in scientific research.

See 5-HT receptor and SB-399885

SB-699551

SB-699551 is a drug which was the first compound developed to act as a selective antagonist for the serotonin receptor 5-HT5A, with selectivity of around 100x over other serotonin receptor subtypes.

See 5-HT receptor and SB-699551

Second messenger system

Second messengers are intracellular signaling molecules released by the cell in response to exposure to extracellular signaling molecules—the first messengers.

See 5-HT receptor and Second messenger system

Serotonin

Serotonin or 5-hydroxytryptamine (5-HT) is a monoamine neurotransmitter.

See 5-HT receptor and Serotonin

Serotonin antagonist and reuptake inhibitor

Serotonin antagonist and reuptake inhibitors (SARIs) are a class of drugs used mainly as antidepressants, but also as anxiolytics and hypnotics.

See 5-HT receptor and Serotonin antagonist and reuptake inhibitor

Serotonin syndrome

Serotonin syndrome (SS) is a group of symptoms that may occur with the use of certain serotonergic medications or drugs.

See 5-HT receptor and Serotonin syndrome

Smooth muscle

Smooth (soft) muscle is one of the three major types of vertebrate muscle tissue, the other being skeletal and cardiac muscle.

See 5-HT receptor and Smooth muscle

Sodium

Sodium is a chemical element; it has symbol Na (from Neo-Latin natrium) and atomic number 11.

See 5-HT receptor and Sodium

Substance P

Substance P (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) and a type of neuropeptide, belonging to the tachykinin family of neuropeptides. It acts as a neurotransmitter and a neuromodulator. Substance P and the closely related neurokinin A (NKA) are produced from a polyprotein precursor after alternative splicing of the preprotachykinin A gene.

See 5-HT receptor and Substance P

Sumatriptan

Sumatriptan, sold under the brand name Imitrex among others, is a medication used to treat migraine headaches and cluster headaches.

See 5-HT receptor and Sumatriptan

Tandospirone

Tandospirone, sold under the brand name Sediel, is an anxiolytic and antidepressant medication used in Japan and China, where it is marketed by Dainippon Sumitomo Pharma.

See 5-HT receptor and Tandospirone

Tegaserod

Tegaserod is a 5-HT4 agonist manufactured by Novartis and sold under the names Zelnorm and Zelmac for the management of irritable bowel syndrome and constipation.

See 5-HT receptor and Tegaserod

Thermoregulation

Thermoregulation is the ability of an organism to keep its body temperature within certain boundaries, even when the surrounding temperature is very different.

See 5-HT receptor and Thermoregulation

Tramadol

Tramadol, sold under the brand name Ultram among others, is an opioid pain medication and a serotonin–norepinephrine reuptake inhibitor (SNRI) used to treat moderately severe pain.

See 5-HT receptor and Tramadol

Trazodone

Trazodone, sold under many brand names, is an antidepressant medication.

See 5-HT receptor and Trazodone

Trifluoromethylphenylpiperazine

3-Trifluoromethylphenylpiperazine (TFMPP) is a recreational drug of the phenylpiperazine chemical class and is a substituted piperazine.

See 5-HT receptor and Trifluoromethylphenylpiperazine

Triptan

Triptans are a family of tryptamine-based drugs used as abortive medication in the treatment of migraines and cluster headaches.

See 5-HT receptor and Triptan

Tropisetron

Tropisetron is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic to treat nausea and vomiting following chemotherapy, although it has been used experimentally as an analgesic in cases of fibromyalgia.

See 5-HT receptor and Tropisetron

Valerenic acid

Valerenic acid is a sesquiterpenoid constituent of the essential oil of the valerian plant.

See 5-HT receptor and Valerenic acid

Vasopressin

Human vasopressin, also called antidiuretic hormone (ADH), arginine vasopressin (AVP) or argipressin, is a hormone synthesized from the AVP gene as a peptide prohormone in neurons in the hypothalamus, and is converted to AVP.

See 5-HT receptor and Vasopressin

Vilazodone

Vilazodone, sold under the brand name Viibryd among others, is a medication used to treat major depressive disorder.

See 5-HT receptor and Vilazodone

Vortioxetine

Vortioxetine, sold under the brand name Brintellix among others, is an antidepressant of the serotonin modulator and stimulator (SMS) class.

See 5-HT receptor and Vortioxetine

WAY-100135

WAY-100135 is a serotonergic drug of the phenylpiperazine family which is used in scientific research.

See 5-HT receptor and WAY-100135

WAY-100635

WAY-100635 is a piperazine drug and research chemical widely used in scientific studies.

See 5-HT receptor and WAY-100635

WAY-181187

WAY-181187 is a high affinity and selective 5-HT6 receptor full agonist.

See 5-HT receptor and WAY-181187

WAY-208466

WAY-208466 is a potent and highly selective full agonist of the 5-HT6 receptor.

See 5-HT receptor and WAY-208466

YM-348

YM-348 is an indazole derivative drug which acts as a potent and selective 5-HT2C receptor agonist, with an EC50 of 1nM and 15x selectivity over 5-HT2A, although it only has moderate selectivity of 3x over the closely related 5-HT2B receptor.

See 5-HT receptor and YM-348

Yohimbine

Yohimbine, also known as quebrachine, is an indole alkaloid derived from the bark of the African tree Pausinystalia johimbe; also from the bark of the unrelated South American tree Aspidosperma quebracho-blanco.

See 5-HT receptor and Yohimbine

Zacopride

Zacopride is a potent antagonist at the 5-HT3 receptor and an agonist at the 5-HT4 receptor.

See 5-HT receptor and Zacopride

Ziprasidone

Ziprasidone, sold under the brand name Geodon among others, is an atypical antipsychotic used to treat schizophrenia and bipolar disorder.

See 5-HT receptor and Ziprasidone

Zolmitriptan

Zolmitriptan, sold under the brand name Zomig among others, is a triptan used in the acute treatment of migraine attacks with or without aura and cluster headaches.

See 5-HT receptor and Zolmitriptan

1-(2-Diphenyl)piperazine

1-(2-Diphenyl)piperazine, also known as RA-7, is a drug which acts as a potent and selective antagonist at the 7 serotonin receptor.

See 5-HT receptor and 1-(2-Diphenyl)piperazine

2,5-Dimethoxy-4-methylamphetamine

2,5-Dimethoxy-4-methylamphetamine (DOM; known as STP, standing for "Serenity, Tranquility and Peace") is a psychedelic and a substituted amphetamine.

See 5-HT receptor and 2,5-Dimethoxy-4-methylamphetamine

2-Methyl-5-hydroxytryptamine

2-Methyl-5-hydroxytryptamine (2-Methylserotonin, 2-Methyl-5-HT) is a tryptamine derivative closely related to the neurotransmitter serotonin which acts as a moderately selective full agonist at the 5-HT3 receptor.

See 5-HT receptor and 2-Methyl-5-hydroxytryptamine

25I-NBOMe

25I-NBOMe (2C-I-NBOMe, Cimbi-5, and also shortened to "25I"), also known as Smiles, or N-Bomb, is a novel synthetic psychoactive substance with strong hallucinogenic properties, synthesized in 2003 for research purposes.

See 5-HT receptor and 25I-NBOMe

2C-B

2C-B (4-bromo-2,5-dimethoxyphenethylamine), also known as Nexus, is a synthetic psychedelic drug of the 2C family, mainly used as a recreational drug.

See 5-HT receptor and 2C-B

5-Carboxamidotryptamine

5-Carboxamidotryptamine (5-CT) is a tryptamine derivative closely related to the neurotransmitter serotonin.

See 5-HT receptor and 5-Carboxamidotryptamine

5-HT1 receptor

The 5-HT1 receptors are a subfamily of the 5-HT serotonin receptors that bind to the endogenous neurotransmitter serotonin (also known as 5-hydroxytryptamine, or 5-HT). 5-HT receptor and 5-HT1 receptor are serotonin receptors.

See 5-HT receptor and 5-HT1 receptor

5-HT1A receptor

The serotonin 1A receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter. 5-HT receptor and 5-HT1A receptor are serotonin receptors.

See 5-HT receptor and 5-HT1A receptor

5-HT1B receptor

5-hydroxytryptamine receptor 1B also known as the 5-HT1B receptor is a protein that in humans is encoded by the HTR1B gene. 5-HT receptor and 5-HT1B receptor are serotonin receptors.

See 5-HT receptor and 5-HT1B receptor

5-HT1D receptor

5-hydroxytryptamine (serotonin) receptor 1D, also known as HTR1D, is a 5-HT receptor, but also denotes the human gene encoding it. 5-HT receptor and 5-HT1D receptor are serotonin receptors.

See 5-HT receptor and 5-HT1D receptor

5-HT1E receptor

5-hydroxytryptamine (serotonin) 1E receptor (5-HT1E) is a highly expressed human G-protein coupled receptor that belongs to the 5-HT1 receptor family (Gi-coupled serotonin receptor). 5-HT receptor and 5-HT1E receptor are serotonin receptors.

See 5-HT receptor and 5-HT1E receptor

5-HT1F receptor

5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it. 5-HT receptor and 5-HT1F receptor are serotonin receptors.

See 5-HT receptor and 5-HT1F receptor

5-HT2 receptor

The 5-HT2 receptors are a subfamily of 5-HT receptors that bind the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). 5-HT receptor and 5-HT2 receptor are serotonin receptors.

See 5-HT receptor and 5-HT2 receptor

5-HT2A receptor

The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). 5-HT receptor and 5-HT2A receptor are serotonin receptors.

See 5-HT receptor and 5-HT2A receptor

5-HT2B receptor

5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT receptor and 5-HT2B receptor are serotonin receptors.

See 5-HT receptor and 5-HT2B receptor

5-HT2C receptor

The 5-HT2C receptor is a subtype of the 5-HT2 receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). 5-HT receptor and 5-HT2C receptor are serotonin receptors.

See 5-HT receptor and 5-HT2C receptor

5-HT3 receptor

The 5-HT3 receptor belongs to the Cys-loop superfamily of ligand-gated ion channels (LGICs) and therefore differs structurally and functionally from all other 5-HT receptors (5-hydroxytryptamine, or serotonin receptors) which are G protein-coupled receptors. 5-HT receptor and 5-HT3 receptor are serotonin receptors.

See 5-HT receptor and 5-HT3 receptor

5-HT4 receptor

5-Hydroxytryptamine receptor 4 is a protein that in humans is encoded by the HTR4 gene. 5-HT receptor and 5-HT4 receptor are serotonin receptors.

See 5-HT receptor and 5-HT4 receptor

5-HT5A receptor

5-Hydroxytryptamine (serotonin) receptor 5A, also known as HTR5A, is a protein that in humans is encoded by the HTR5A gene. 5-HT receptor and 5-HT5A receptor are serotonin receptors.

See 5-HT receptor and 5-HT5A receptor

5-HT5B receptor

5-HT5B receptor is a 5-HT receptor protein and the gene which encodes it. 5-HT receptor and 5-HT5B receptor are serotonin receptors.

See 5-HT receptor and 5-HT5B receptor

5-HT6 receptor

The 5HT6 receptor is a subtype of 5HT receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5HT). 5-HT receptor and 5-HT6 receptor are serotonin receptors.

See 5-HT receptor and 5-HT6 receptor

5-HT7 receptor

The 5-HT7 receptor is a member of the GPCR superfamily of cell surface receptors and is activated by the neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). 5-HT receptor and 5-HT7 receptor are serotonin receptors.

See 5-HT receptor and 5-HT7 receptor

5-MeO-DMT

5-MeO-DMT (5-methoxy-N,N-dimethyltryptamine) or O-methyl-bufotenin is a psychedelic of the tryptamine class.

See 5-HT receptor and 5-MeO-DMT

5-Methoxytryptamine

5-Methoxytryptamine (5-MT), also known as mexamine, is a tryptamine derivative closely related to the neurotransmitters serotonin and melatonin.

See 5-HT receptor and 5-Methoxytryptamine

6-APB

6-APB (6-(2-aminopropyl)benzofuran) is an empathogenic psychoactive compound of the substituted benzofuran and substituted phenethylamine classes.

See 5-HT receptor and 6-APB

8-OH-DPAT

8-OH-DPAT is a research chemical of the aminotetralin chemical class which was developed in the 1980s and has been widely used to study the function of the 5-HT1A receptor.

See 5-HT receptor and 8-OH-DPAT

See also

Serotonin receptors

References

[1] https://en.wikipedia.org/wiki/5-HT_receptor

Also known as 5-HT receptor 4, 5-HT receptors, 5-HT1 like, 5-Hydroxytryptamine receptor, 5-carboxytryptamine, 5-ct, 5HT receptor, 5HT-3 receptor, 5HT-4 receptor, 5ht-receptor, 5ht-receptors, 5ht4, 5htr, Receptors, serotonin, Serotonin plasma membrane transport proteins, Serotonin r, Serotonin receptor, Serotonin receptors.

, CP-93129, CP-94253, Cyanopindolol, Cyclic adenosine monophosphate, Cyproheptadine, Dazopride, Depolarization, Diglyceride, Dihydroergotamine, Dolasetron, Dopamine, Doxepin, E-55888, E-6837, EGIS-12,233, Eletriptan, Eltoprazine, EMD-386088, EMDT, Empathogen, Eplivanserin, Ergometrine, Ergotamine, Etoperidone, F-15,599, Fenfluramine, Flesinoxan, Fluoxetine, Frovatriptan, G protein-coupled receptor, GABA, Gastrointestinal tract, Gepirone, Gi alpha subunit, Glossary of biology, Glutamic acid, Gq alpha subunit, GR-127935, Granisetron, Gs alpha subunit, Hallucinogen, Haloperidol, Heteroreceptor, Hydroxyzine, Hypnotic, Iloperidone, Imipramine, Inositol trisphosphate, Iodocyanopindolol, Ion channel, Ipsapirone, Isamoltane, Ketanserin, Lasmiditan, Latrepirdine, Lecozotan, Ligand (biochemistry), Ligand-gated ion channel, Lisuride, Lorcaserin, LSD, LY-334370, Lysine, MDMA, Mefway (18F), Memantine, Mescaline, Metergoline, Methylergometrine, Methylphenidate, Methysergide, Metitepine, Metoclopramide, Mianserin, Migraine, Mirtazapine, Mood (psychology), Mosapride, MS-245, NAN-190, Naratriptan, Nebivolol, Nefazodone, Nematode, Neurotransmission, Neurotransmitter, Nootropic, Noradrenergic and specific serotonergic antidepressant, Norepinephrine, Norfenfluramine, Olanzapine, Ondansetron, Oxprenolol, Oxytocin, Paroxetine, Partial agonist, Peripheral nervous system, Piboserod, Pieris rapae, Pimavanserin, Pindolol, Pizotifen, Platelet, PNU-22394, Potassium, Prokinetic agent, Prolactin, Propranolol, Protein Data Bank, Prucalopride, Pseudogene, Psilocin, Psilocybin, Psychedelic drug, Quetiapine, Quipazine, Rauwolscine, Receptor antagonist, Renzapride, Risperidone, Ritanserin, Rizatriptan, Ro 04-6790, Ro60-0175, RS-127445, RS-56812, RS-67,333, RU-24,969, SB-216641, SB-242084, SB-258585, SB-269970, SB-271046, SB-357134, SB-399885, SB-699551, Second messenger system, Serotonin, Serotonin antagonist and reuptake inhibitor, Serotonin syndrome, Smooth muscle, Sodium, Substance P, Sumatriptan, Tandospirone, Tegaserod, Thermoregulation, Tramadol, Trazodone, Trifluoromethylphenylpiperazine, Triptan, Tropisetron, Valerenic acid, Vasopressin, Vilazodone, Vortioxetine, WAY-100135, WAY-100635, WAY-181187, WAY-208466, YM-348, Yohimbine, Zacopride, Ziprasidone, Zolmitriptan, 1-(2-Diphenyl)piperazine, 2,5-Dimethoxy-4-methylamphetamine, 2-Methyl-5-hydroxytryptamine, 25I-NBOMe, 2C-B, 5-Carboxamidotryptamine, 5-HT1 receptor, 5-HT1A receptor, 5-HT1B receptor, 5-HT1D receptor, 5-HT1E receptor, 5-HT1F receptor, 5-HT2 receptor, 5-HT2A receptor, 5-HT2B receptor, 5-HT2C receptor, 5-HT3 receptor, 5-HT4 receptor, 5-HT5A receptor, 5-HT5B receptor, 5-HT6 receptor, 5-HT7 receptor, 5-MeO-DMT, 5-Methoxytryptamine, 6-APB, 8-OH-DPAT.