Acetryptine

Acetryptine (INN) (developmental code name W-2965-A), also known as 5-acetyltryptamine (5-AT), is a drug described as an antihypertensive agent which was never marketed. ^[1]

25 relations: Antihypertensive drug, Azepindole, Drug, Enzyme inhibitor, Indorenate, International nonproprietary name, Ligand (biochemistry), Metralindole, Monoamine oxidase A, Monoamine oxidase inhibitor, Pargyline, Pirlindole, Receptor (biochemistry), Serotonin, Substituted tryptamine, Sumatriptan, Tetrindole, 5-(Nonyloxy)tryptamine, 5-Benzyloxytryptamine, 5-Carboxamidotryptamine, 5-Ethoxy-DMT, 5-HT receptor, 5-HT1A receptor, 5-HT1D receptor, 5-Methoxytryptamine.

Antihypertensive drug

Antihypertensives are a class of drugs that are used to treat hypertension (high blood pressure). Acetryptine and Antihypertensive drug are antihypertensive agents.

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Azepindole (McN-2453) is a tricyclic compound with antidepressant and antihypertensive effects that was developed in the late 1960s but was never marketed. Acetryptine and Azepindole are antihypertensive agent stubs.

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Drug

A drug is any chemical substance other than a nutrient or an essential dietary ingredient, which, when administered to a living organism, produces a biological effect.

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Enzyme inhibitor

An enzyme inhibitor is a molecule that binds to an enzyme and blocks its activity.

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Indorenate

Indorenate (TR-3369), is a tryptamine derivative which acts as an agonist at the 5-HT1A, 5-HT1B and 5-HT2C serotonin receptors. Acetryptine and Indorenate are serotonin receptor agonists.

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International nonproprietary name

An international nonproprietary name (INN) is an official generic and nonproprietary name given to a pharmaceutical drug or an active ingredient.

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Ligand (biochemistry)

In biochemistry and pharmacology, a ligand is a substance that forms a complex with a biomolecule to serve a biological purpose.

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Metralindole

Metralindole (Inkazan) is a reversible inhibitor of monoamine oxidase A (RIMA) which was investigated in Russia as a potential antidepressant. Acetryptine and Metralindole are tryptamines.

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Monoamine oxidase A

Monoamine oxidase A, also known as MAO-A, is an enzyme (E.C. 1.4.3.4) that in humans is encoded by the MAOA gene.

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Monoamine oxidase inhibitor

Monoamine oxidase inhibitors (MAOIs) are a class of drugs that inhibit the activity of one or both monoamine oxidase enzymes: monoamine oxidase A (MAO-A) and monoamine oxidase B (MAO-B).

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Pargyline

Pargyline (brand name Eutonyl) is an irreversible selective monoamine oxidase (MAO)-B inhibitor drug (IC50 for MAO-A is 11.52 nM and for MAO-B is 8.20 nM) It was brought to market in the US and the UK by Abbott in 1963 as an antihypertensive drug branded "Eutonyl". Acetryptine and Pargyline are antihypertensive agent stubs and antihypertensive agents.

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Pirlindole

Pirlindole (Lifril, Pyrazidol) is mainly a reversible inhibitor of monoamine oxidase A (RIMA) and secondly a SNRI which was developed and is used in Russia as an antidepressant.

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Receptor (biochemistry)

In biochemistry and pharmacology, receptors are chemical structures, composed of protein, that receive and transduce signals that may be integrated into biological systems.

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Serotonin

Serotonin or 5-hydroxytryptamine (5-HT) is a monoamine neurotransmitter.

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Substituted tryptamine

Substituted tryptamines, or serotonin analogues, are organic compounds which may be thought of as being derived from tryptamine itself. Acetryptine and Substituted tryptamine are tryptamines.

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Sumatriptan

Sumatriptan, sold under the brand name Imitrex among others, is a medication used to treat migraine headaches and cluster headaches.

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Tetrindole

Tetrindole was a drug candidate that functions by reversibly inhibiting monoamine oxidase A; it was first synthesized in Moscow in the early 1990s.

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5-(Nonyloxy)tryptamine

5-(Nonyloxy)tryptamine is a tryptamine derivative which acts as a selective agonist at the 5-HT1B receptor. Acetryptine and 5-(Nonyloxy)tryptamine are serotonin receptor agonists and tryptamines.

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5-Benzyloxytryptamine

5-Benzyloxytryptamine (5-BT), is a tryptamine derivative which acts as an agonist at the 5-HT1D, 5-HT2 and 5-HT6 serotonin receptors, and an antagonist of TRPM8. Acetryptine and 5-Benzyloxytryptamine are serotonin receptor agonists and tryptamines.

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5-Carboxamidotryptamine

5-Carboxamidotryptamine (5-CT) is a tryptamine derivative closely related to the neurotransmitter serotonin. Acetryptine and 5-Carboxamidotryptamine are serotonin receptor agonists and tryptamines.

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5-Ethoxy-DMT

5-Ethoxy-DMT (5-ethoxy-N,N-dimethyltryptamine, 5-EtO-DMT, O-ethylbufotenine) is a tryptamine derivative which has been previously synthesized as a chemical intermediate, but has not been studied to determine its pharmacology. Acetryptine and 5-Ethoxy-DMT are tryptamines.

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5-HT receptor

5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in the central and peripheral nervous systems.

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5-HT1A receptor

The serotonin 1A receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter.

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5-HT1D receptor

5-hydroxytryptamine (serotonin) receptor 1D, also known as HTR1D, is a 5-HT receptor, but also denotes the human gene encoding it.

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5-Methoxytryptamine

5-Methoxytryptamine (5-MT), also known as mexamine, is a tryptamine derivative closely related to the neurotransmitters serotonin and melatonin. Acetryptine and 5-Methoxytryptamine are serotonin receptor agonists.

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References

[1] https://en.wikipedia.org/wiki/Acetryptine

Also known as 5-Acetyl-tryptamine, 5-Acetyltryptamine, Acetriptin, Acetriptina, Acetriptine, Acetriptinum, Acetryptin, Acetryptina, Acetryptinum, W 2965-A, W 2965A, W-2965 A, W-2965-A, W-2965A, W2965 A, W2965-A, W2965A.

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Acetryptine

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