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75 relations: Adrenorphin, Agonist-antagonist, Akuammicine, Anorexia nervosa, AP-237, Arrestin beta 1, Beta-2 adrenergic receptor, Biphalin, BU-48, BW373U86, C-8813, CERC-501, Coronaridine, CR665, Cyclazocine, Cyprodime, DADLE, DAMGO, Desmethylclozapine, Dextrallorphan, Dezocine, Dihydromorphine, Dor, DPI-221, DPI-287, DPI-3290, Enkephalin, Etorphine, G protein-coupled inwardly-rectifying potassium channel, Gi alpha subunit, GPRASP1, Hallucination, Hemorphin-4, Heroin, Hydrocodone/paracetamol, Hypericum perforatum, Incarvillateine, Index of biochemistry articles, Ischemic preconditioning, Κ-opioid receptor, Μ-opioid receptor, JDTic, Ketamine, Leu-enkephalin, MCOPPB, Met-enkephalin, Mitragynine pseudoindoxyl, Morphiceptin, N-2′-Indolylnaltrexamine, N-Phenethyl-14-ethoxymetopon, ..., Naltriben, Naltrindole, Neurotransmitter, Nociceptin receptor, Norbinaltorphimine, Norbuprenorphine, Opioid, Penicillium parvum, Proglumide, RB-101, Rhodopsin-like receptors, RWJ-394674, SC-17599, Sigma receptor, SNC-80, SoRI-9409, Spiradoline, TAN-67, Tonazocine, Trevena Inc, U-77891, 18,19-Dehydrobuprenorphine, 18-Methylaminocoronaridine, 25I-NBOMe, 7-Spiroindanyloxymorphone. Expand index (25 more) »
Adrenorphin
Adrenorphin, also sometimes referred to as metorphamide, is an endogenous, C-terminally amidated, opioid octapeptide (Tyr-Gly-Gly-Phe-Met-Arg-Arg-Val-NH2) that is produced from proteolytic cleavage of proenkephalin A and is widely distributed throughout the mammalian brain.
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Agonist-antagonist
In pharmacology the term agonist-antagonist or mixed agonist/antagonist is used to refer to a drug which under some conditions behaves as an agonist (a substance that fully activates the receptor that it binds to) while under other conditions, behaves as an antagonist (a substance that binds to a receptor but does not activate and can block the activity of other agonists).
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Akuammicine
Akuammicine is an alkaloid found in Vinca minor and Aspidosperma.
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Anorexia nervosa
Anorexia nervosa, often referred to simply as anorexia, is an eating disorder characterized by low weight, fear of gaining weight, and a strong desire to be thin, resulting in food restriction.
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AP-237
AP-237 (1-butyryl-4-cinnamylpiperazine) is an opioid analgesic drug that was widely used in China to treat pain in cancer patients as of 1986.
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Arrestin beta 1
Arrestin, beta 1, also known as ARRB1, is a protein which in humans is encoded by the ARRB1 gene.
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Beta-2 adrenergic receptor
The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that interacts with (binds) epinephrine, a hormone and neurotransmitter (ligand synonym, adrenaline) whose signaling, via a downstream L-type calcium channel interaction, mediates physiologic responses such as smooth muscle relaxation and bronchodilation.
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Biphalin
Biphalin is a dimeric enkephalin endogenous peptide (Tyr-D-Ala-Gly-Phe-NH)2 composed of two tetrapeptides derived from enkephalins, connected 'tail-to-tail' by a hydrazide bridge.
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BU-48
BU-48 is a drug that is used in scientific research.
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BW373U86
(+)-BW373U86 is an opioid analgesic drug used in scientific research.
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C-8813
C-8813 (thiobromadol) is a potent μ-opioid receptor agonist with a distinctive chemical structure which is not closely related to other established families of opioid drugs.
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CERC-501
CERC-501 (originally known as LY-2456302) is a selective antagonist of the κ-opioid receptor (KOR) which was originally developed by Eli Lilly and is now under development by Janssen Pharmaceuticals for the treatment of major depressive disorder and substance use disorders including alcoholism, nicotine addiction, and illicit drug dependence.
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Coronaridine
Coronaridine, also known as 18-carbomethoxyibogamine, is an alkaloid found in Tabernanthe iboga and related species, including Tabernaemontana divaricata for which (under the now obsolete synonym Ervatamia coronaria) it was named.
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CR665
CR665 (H-D-Phe-D-Phe-D-Nle-D-Arg-NH-4-Picolyl), also known by the previous developmental code names FE-200665 and JNJ-38488502, is an all D-amino acid peptide that acts as a peripherally restricted κ-opioid receptor agonist.
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Cyclazocine
Cyclazocine is a mixed opioid agonist/antagonist related to dezocine, pentazocine and phenazocine.
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Cyprodime
Cyprodime is an opioid antagonist from the morphinan family of drugs.
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DADLE
DADLE (-Enkephalin) is a synthetic opioid peptide with analgesic properties.
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DAMGO
DAMGO (-enkephalin) is a synthetic opioid peptide with high μ-opioid receptor specificity.
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Desmethylclozapine
N-Desmethylclozapine (NDMC), or norclozapine, is a major active metabolite of the atypical antipsychotic drug clozapine.
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Dextrallorphan
Dextrallorphan (DXA) is an opioid derivative chemical of the morphinan class that is used in scientific research.
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Dezocine
Dezocine (INN, USAN) (brand name Dalgan) is a marketed opioid analgesic of the benzomorphan group.
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Dihydromorphine
Dihydromorphine (Paramorfan, Paramorphan) is a semi-synthetic opioid structurally related to and derived from morphine.
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Dor
DOR or Dor or DoR may refer to.
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DPI-221
DPI-221 is a opioid drug that is used in scientific research.
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DPI-287
DPI-287 is an opioid drug that is used in scientific research.
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DPI-3290
DPI-3290 was discovered by scientists at Burroughs Wellcome and licensed to Delta Pharmaceutical and is a drug that is used in scientific research.
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Enkephalin
An enkephalin (occasionally spelled encephalin) is a pentapeptide involved in regulating nociception in the body.
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Etorphine
Etorphine (M99) is a semi-synthetic opioid possessing an analgesic potency approximately 1,000–3,000 times that of morphine.
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G protein-coupled inwardly-rectifying potassium channel
The G protein-coupled inwardly-rectifying potassium channels (GIRKs) are a family of inward-rectifier potassium ion channels which are activated (opened) via a signal transduction cascade starting with ligand-stimulated G protein-coupled receptors (GPCRs).
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Gi alpha subunit
Gi alpha subunit (Gαi, or Gi/G0 or Gi protein) is a heterotrimeric G protein subunit that inhibits the production of cAMP from ATP.
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GPRASP1
G-protein coupled receptor-associated sorting protein 1 is a protein that in humans is encoded by the GPRASP1 gene.
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Hallucination
A hallucination is a perception in the absence of external stimulus that has qualities of real perception.
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Hemorphin-4
Hemorphin-4 is an endogenous opioid peptide of the hemorphin family which possesses antinociceptive properties and is derived from the β-chain of hemoglobin in the bloodstream.
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Heroin
Heroin, also known as diamorphine among other names, is an opioid most commonly used as a recreational drug for its euphoric effects.
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Hydrocodone/paracetamol
Hydrocodone/paracetamol, also known as hydrocodone/acetaminophen or hydrocodone/APAP and marketed under the trade name Vicodin and Norco among others, is the combination of an opioid pain medication, hydrocodone, with paracetamol (acetaminophen).
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Hypericum perforatum
Hypericum perforatum, known as perforate St John's-wort, common Saint John's wort and St John's wort, is a flowering plant in the family Hypericaceae.
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Incarvillateine
Incarvillateine is a complex monoterpene alkaloid that is a derivative of α-truxillic acid.
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Index of biochemistry articles
Biochemistry is the study of the chemical processes in living organisms.
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Ischemic preconditioning
Ischemic preconditioning (IPC) is an experimental technique for producing resistance to the loss of blood supply, and thus oxygen, to tissues of many types.
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Κ-opioid receptor
The κ-opioid receptor (KOR) is a G protein-coupled receptor that in humans is encoded by the OPRK1 gene.
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Μ-opioid receptor
The μ-opioid receptors (MOR) are a class of opioid receptors with a high affinity for enkephalins and beta-endorphin, but a low affinity for dynorphins.
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JDTic
JDTic is a selective, long-acting ("inactivating") antagonist of the κ-opioid receptor (KOR).
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Ketamine
Ketamine, sold under the brand name Ketalar among others, is a medication mainly used for starting and maintaining anesthesia.
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Leu-enkephalin
Leu-enkephalin is an endogenous opioid peptide neurotransmitter with the amino acid sequence Tyr-Gly-Gly-Phe-Leu that is found naturally in the brains of many animals, including humans.
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MCOPPB
MCOPPB is a drug which acts as a potent and selective agonist for the nociceptin receptor, with a pKi of 10.07 and much weaker activity at other opioid receptors.
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Met-enkephalin
Met-enkephalin, also known as metenkefalin (INN), sometimes referred to as opioid growth factor (OGF), is a naturally occurring, endogenous opioid peptide that has opioid effects of a relatively short duration.
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Mitragynine pseudoindoxyl
Mitragynine pseudoindoxyl is a rearrangement product of 7-hydroxymitragynine.
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Morphiceptin
Morphiceptin is a tetrapeptide (Tyr-Pro-Phe-Pro-NH2) that is a selective μ-opioid receptor agonist.
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N-2′-Indolylnaltrexamine
N-2′-Indolylnaltrexamine (INTA) is an opioid and derivative of β-naltrexamine.
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N-Phenethyl-14-ethoxymetopon
N-Phenethyl-14-ethoxymetopon is a drug that is a derivative of metopon.
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Naltriben
Naltriben is a potent and selective antagonist for the delta opioid receptor, which is used in scientific research.
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Naltrindole
Naltrindole is a highly potent, highly selective delta opioid receptor antagonist used in biomedical research.
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Neurotransmitter
Neurotransmitters are endogenous chemicals that enable neurotransmission.
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Nociceptin receptor
The nociceptin opioid peptide receptor (NOP), also known as the nociceptin/orphanin FQ (N/OFQ) receptor or kappa-type 3 opioid receptor, is a protein that in humans is encoded by the OPRL1 (opioid receptor-like 1) gene.
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Norbinaltorphimine
Norbinaltorphimine (nor-BNI or nBNI) is an opioid antagonist used in scientific research.
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Norbuprenorphine
Norbuprenorphine is a major active metabolite of the opioid modulator buprenorphine.
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Opioid
Opioids are substances that act on opioid receptors to produce morphine-like effects.
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Penicillium parvum
Penicillium parvum is an anamorph species of the genus of Penicillium which was isolated from soil in Papua New Guinea.
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Proglumide
Proglumide (Milid) is a drug that inhibits gastrointestinal motility and reduces gastric secretions.
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RB-101
RB-101 is a drug that acts as an enkephalinase inhibitor, which is used in scientific research.
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Rhodopsin-like receptors
Rhodopsin-like receptors are a family of proteins that comprise the largest group of G protein-coupled receptors.
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RWJ-394674
RWJ-394674 is a drug that is used in scientific research.
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SC-17599
SC-17599 is a steroid derivative drug discovered in 1968 which acts as a selective μ-opioid receptor agonist, with little or no affinity for the δ-opioid or κ-opioid receptors.
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Sigma receptor
Schematic σ receptor The sigma receptors σ1 and σ2 bind to ligands such as 4-PPBP (4-phenyl-1-(4-phenylbutyl) piperidine), SA 4503 (cutamesine), ditolylguanidine, dimethyltryptamine, and siramesine.
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SNC-80
SNC-80 is an opioid analgesic drug that selectively activates μ–δ opioid receptor heteromers and is used in scientific research.
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SoRI-9409
SoRI-9409 is a mixed mu opioid receptor partial agonist and delta opioid receptor antagonist, used in biomedical research.
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Spiradoline
Spiradoline (U-62066) is a drug which acts as a highly selective κ-opioid agonist.
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TAN-67
TAN-67 (SB-205,607) is a opioid drug used in scientific research that acts as a potent and selective δ-opioid agonist, selective for the δ1 subtype.
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Tonazocine
Tonazocine (WIN-42,156) is an opioid analgesic of the benzomorphan family which made it to phase II clinical trials for the treatment of postoperative pain, but development was apparently ceased and ultimately it was never marketed.
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Trevena Inc
Trevena Inc is a clinical stage biopharmaceutical company, headquartered in Chesterbrook, Pennsylvania, USA, and is involved in the discovery and development of G-protein coupled receptors (GPCR) biased ligands.
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U-77891
U-77891 is an opioid analgesic drug that was first synthesized in 1983 by the Upjohn company.
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18,19-Dehydrobuprenorphine
18,19-Dehydrobuprenorphine (HS-599) is a derivative of buprenorphine.
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18-Methylaminocoronaridine
(–)-18-Methylaminocoronaridine (18-MAC) is a second generation synthetic derivative of ibogaine developed by the research team led by the pharmacologist Stanley D. Glick from the Albany Medical College and the chemist Martin E. Kuehne from the University of Vermont.
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25I-NBOMe
25I-NBOMe (2C-I-NBOMe, Cimbi-5, also shortened to "25I") is a psychedelic hallucinogen that is used in biochemistry research for mapping the brains usage of the type 2A serotonin receptor and later also has been used for recreational purpose.
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7-Spiroindanyloxymorphone
7-Spiroindanyloxymorphone (SIOM) is a drug that is used in scientific research. It is a selective δ-opioid agonist. It is a derivative of oxymorphone.
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D-Opioid, D-Opioid receptor, D-opioid, D-opioid receptor, Delta Opioid, Delta Opioid receptor, Delta opioid, Delta opioid receptor, Delta-Opioid, Delta-Opioid receptor, Delta-opioid, Delta-opioid receptor, OPRD1, OPRD1 (gene).
References
[1] https://en.wikipedia.org/wiki/Δ-opioid_receptor
